Multidrug Resistance-associated Protein 2 - MRP2 Inhibitors

MRP2 Inhibitors

Drug Class Indications Source Structure
probenecid uricosuric gout
hyperuricemia
furosemide loop diuretic heart failure
edema
ritonavir protease inhibitor antiretroviral
saquinavir protease inhibitor antiretroviral
lamivudine Nucleoside analog antiviral
abacavir Nucleoside analog antiretroviral
emtricitabine Nucleoside analog antiviral
efavirenz NNRTI antiretroviral
delavirdine NNRTI antiretroviral
nevirapine NNRTI antiretroviral
cidofovir nucleoside phosphonate antiviral
adefovir nucleoside phosphonate antiviral
tenofovir nucleoside phosphonate antiviral

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