Excitatory Amino Acid Antagonist

An excitatory amino acid antagonist is a pharmacological agent which acts to decrease the stimulation of receptors for excitatory amino acids (primarily glutamate).

Examples include:

  • 2-amino-5-phosphonovalerate
  • dextromethorphan
  • dextrorphan
  • ibogaine
  • ifenprodil
  • ketamine
  • ketobemidone
  • kynurenic acid
  • memantine
  • phencyclidine
  • phenobarbital
  • riluzole